Roach's Introductory Clinical Pharmacology 11th Edition - Cholinergic Blocking Drugs Related

Review Roach's Introductory Clinical Pharmacology 11th Edition - Cholinergic Blocking Drugs related questions and content

When describing the different cholinergic blockers, which of the following would a nursing instructor include as affecting only the muscarinic receptors?

  • A. Darifenacin (Enablex)
  • B. Oxybutynin (Ditropan)
  • C. Benztropine (Cogentin)
  • D. Biperiden (Akineton)
  • E. Tolterodine (Detrol)
Correct Answer: A,B,E

Rationale: Antispasmodic cholinergic blocking drugs, like darifenacin (Enablex), oxybutynin (Ditropan), and tolterodine (Detrol), only affect muscarinic receptors in the parasympathetic nervous system and have no effect on nicotinic receptors.